A Guide to Measuring Drug-Target Residence Time
This guide provides technical background on concepts and techniques for using Transcreener biochemical assays to measure drug-target residence times in a high throughput format.
Download this guide to learn more including
-The basics of residence time and its importance to drug discovery
-A comparison of methods used for residence time determination
-Using the jump-dilution method with Transcreener Assays
-Examples of determining residence time for kinases, phosphodiesterases, and glycosyltransferases
-Measuring residence time in an HTS compatible format